Palladium-Catalyzed Direct Arylation of Imidazolone N-Oxides with Aryl Bromides and Its Application in the Synthesis of GSK2137305
Author:
Affiliation:
1. Medicinal Chemistry Department, AMRI, 26 Corporate Circle, P.O. Box 15098, Albany, New York 12212-5098, United States
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/ol300468g
Reference56 articles.
1. Kottamides A−D: Novel Bioactive Imidazolone-Containing Alkaloids from the New Zealand Ascidian Pycnoclavella kottae
2. An Efficient and Scalable Synthesis of the Spirocyclic Glycine Transporter Inhibitor GSK2137305
3. Completely N1-Selective Palladium-Catalyzed Arylation of Unsymmetric Imidazoles: Application to the Synthesis of Nilotinib
4. cBlunt, R.; Cooper, D. G.; Porter, R. A.WO 2009034061, 2009.
5. dAhmad, N. M.; Lai, J. Y. Q.; Andreotti, D.WO 2008092876, 2008.
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