Novel and Expeditious Microwave-Assisted Three-Component Reactions for the Synthesis of Spiroimidazolin-4-ones
Author:
Affiliation:
1. ArQule, Incorporated, Division of Chemical Technologies, 19 Presidential Way, Woburn, Massachusetts 01801
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/jo060228q
Reference21 articles.
1. Accelerating lead development by microwave-enhanced medicinal chemistry
2. (b) Leadbeater, N. E.Chem. Commun.2005, 2881 and references therein.
3. Total Synthesis of the Amaryllidaceae Alkaloid (+)-Plicamine and Its Unnatural Enantiomer by Using Solid-Supported Reagents and Scavengers in a Multistep Sequence of Reactions We gratefully acknowledge financial support from Pfizer Central Research for a Postdoctoral Fellowship (to I.R.B.), the BP endowment and the Novartis Research Fellowship (to S.V.L.), and Pharmacia & Upjohn (to C.P.).
4. (a) Bernhart, C. A.; Breliere, J.C.; Clement, J.; Nisato, D.; Perreaut, P. M. EP 454511, 1991; FR 2659967, 1990; US 5270317, 1993; WO 9114679, 1991.
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