Practical, Asymmetric Route to Sitagliptin and Derivatives: Development and Origin of Diastereoselectivity-Reference-Cited by-同舟云学术

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Practical, Asymmetric Route to Sitagliptin and Derivatives: Development and Origin of Diastereoselectivity

Published:2015-03-23 Issue:7 Volume:17 Page:1742-1745
ISSN:1523-7060
Container-title:Organic Letters
language:en
Short-container-title:Org. Lett.

Author:

Gutierrez Osvaldo¹,Metil Dattatray²,Dwivedi Namrata²,Gudimalla Nagaraju²,Chandrashekar E. R. R.²,Dahanukar Vilas H.²,Bhattacharya Apurba²,Bandichhor Rakeshwar²,Kozlowski Marisa C.¹

Affiliation:

1. Roy and Diana Vagelos Laboratories, Department of Chemistry, University of Pennsylvania, 231 South 34th Street, Philadelphia, Pennsylvania 19104 United States

2. API R&D, Integrated Product Development, Dr. Reddy’s Laboratories, Ltd., Innovation Plaza, Bachupally, Qutubullapur, Hyderabad 500090, A.P., India

Funder

National Institute of General Medical Sciences

Dr. Reddy?s Laboratories Ltd.

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.orglett.5b00520

Reference56 articles.

1. Chiral heterocyclic β-enamino esters: convenient synthesis and diastereoselective reduction

2. Asymmetric synthesis with chiral hydrogenolysable amines. Cyclic β-enamino ester reduction a diastereoselective route to 2,3-disubstituted pyrrolidines

3. Chiral cyclic β-amino esters. Part II: Synthesis by diastereoselective reduction of enamino esters

4. Stereocontrolled reduction of chiral pyrrolidine and piperidine β-enamino esters: formal enantioselective synthesis of (+)-calvine

5. Diastereocontrolled reduction of cyclic β-enaminones. A new diastereoselective route to 2,6-disubstituted piperidines

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1. Enantioselective Synthesis of (R)-Sitagliptin via Phase-Transfer Catalytic aza-Michael Addition;ACS Omega;2024-03-21

2. Synthesis of β-Amino Carbonyl 6-(Aminomethyl)- and 6-(Hydroxymethyl)pyrazolopyrimidines for DPP-4 Inhibition Study;Current Medicinal Chemistry;2022-06-14

3. Solvent Dependency in Stereoselective δ‐Lactam Formation of Chiral α‐Fluoromalonate Derivatives: Stereodivergent Synthesis of Heterocycles with Fluorine Containing Stereocenters Adjacent to Tertiary Stereocenters;Advanced Synthesis & Catalysis;2022-01-31

4. Synthesis of (−)‐( R )‐Sitagliptin by Rh I ‐Catalyzed Asymmetric Hydroamination;European Journal of Organic Chemistry;2021-09-23

5. Design, synthesis and biological evaluation of glycolamide, glycinamide, and β-amino carbonyl 1,2,4-triazole derivatives as DPP-4 inhibitors;Bioorganic Chemistry;2021-09

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