Enantioselective Synthesis of (<i>R</i>)-Sitagliptin via Phase-Transfer Catalytic aza-Michael Addition-Reference-Cited by-同舟云学术

Enantioselective Synthesis of (R)-Sitagliptin via Phase-Transfer Catalytic aza-Michael Addition

Published:2024-03-21 Issue:13 Volume:9 Page:15328-15338
ISSN:2470-1343
Container-title:ACS Omega
language:en
Short-container-title:ACS Omega

Author:

Oh Daehyun¹,Lee Jaeyong¹,Yang Sehun¹,Jung So Hyun¹,Kim Mihyun²^ORCID,Lee Geumwoo¹,Park Hyeung-geun¹^ORCID

Affiliation:

1. Research Institute of Pharmaceutical Sciences and College of Pharmacy, Seoul National University, 1 Gwanak-ro, Gwanak-gu, Seoul 08826, Republic of Korea

2. College of Pharmacy, Gachon University, 191 Hambakmoero, Yeonsu-gu, Incheon 21936, Republic of Korea

Funder

National Research Foundation of Korea

Seoul National University

Publisher

American Chemical Society (ACS)

Link

https://pubs.acs.org/doi/pdf/10.1021/acsomega.3c10080

Reference34 articles.

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4. (2R)-4-Oxo-4-[3-(Trifluoromethyl)-5,6-dihydro[1,2,4]triazolo[4,3-a]pyrazin- 7(8H)-yl]-1-(2,4,5-trifluorophenyl)butan-2-amine: A Potent, Orally Active Dipeptidyl Peptidase IV Inhibitor for the Treatment of Type 2 Diabetes

5. Efficient synthesis of sitagliptin phosphate, a novel DPP-IV inhibitor, via a chiral aziridine intermediate

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