Phosphoramidates as Steering Elements for Highly Selective Access to Complementary Imidazo[1,2-a]pyrimidine Isomers-Reference-Cited by-同舟云学术

Phosphoramidates as Steering Elements for Highly Selective Access to Complementary Imidazo[1,2-a]pyrimidine Isomers

Published:2019-11-18 Issue:23 Volume:21 Page:9527-9531
ISSN:1523-7060
Container-title:Organic Letters
language:en
Short-container-title:Org. Lett.

Author:

White Nicholas A.¹^ORCID,Clagg Kyle¹,Sirois Lauren E.¹^ORCID,Mack Kyle A.¹^ORCID,Al-Sayah Mohammad A.²,Nack William A.³,O’Shea Paul D.³,Zhang Haiming¹^ORCID,Gosselin Francis¹^ORCID

Affiliation:

1. Department of Small Molecule Process Chemistry, Genentech, Inc., 1 DNA Way, South San Francisco, California 94080, United States

2. Department of Small Molecule Analytical Chemistry, Genentech, Inc., 1 DNA Way, South San Francisco, California 94080, United States

3. Exemplify BioPharma, 3000 Eastpark Boulevard, Suite 500-A, Cranbury, New Jersey 08512, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.orglett.9b03702

Reference10 articles.

1. A Highly Selective and Specific PET Tracer for Imaging of Tau Pathologies

2. Concise and high-yield synthesis of T808 and T808P for radiosynthesis of [18F]-T808, a PET tau tracer for Alzheimer’s disease

3. Identification of Three Novel Radiotracers for Imaging Aggregated Tau in Alzheimer’s Disease with Positron Emission Tomography

4. Comparative studies on conventional and microwave-assisted synthesis of a series of 2,4-di and 2,3,4-trisubstituted benzimidazo[1,2-a] pyrimidines and their antimicrobial activities

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