Stereochemical Diversity-Oriented Conformational Restriction Strategy. Development of Potent Histamine H3 and/or H4 Receptor Antagonists with an Imidazolylcyclopropane Structure-Reference-Cited by-同舟云学术

Stereochemical Diversity-Oriented Conformational Restriction Strategy. Development of Potent Histamine H3 and/or H4 Receptor Antagonists with an Imidazolylcyclopropane Structure

Published:2006-08-04 Issue:18 Volume:49 Page:5587-5596
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Watanabe Mizuki¹,Kazuta Yuji¹,Hayashi Hideki¹,Yamada Shizuo¹,Matsuda Akira¹,Shuto Satoshi¹

Affiliation:

1. Graduate School of Pharmaceutical Sciences, Hokkaido University, Kita-12, Nishi-6, Kita-ku, Sapporo 060-0812, Japan, and Department of Pharmacokinetics and Pharmacodynamics and COE Program in the 21st Century, School of Pharmaceutical Sciences, University of Shizuoka, 52-1 Yada, Suruga-ku, Shizuoka 422-8526, Japan

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0603318

Reference42 articles.

1. Modelling G-protein-coupled receptors for drug design

2. Crystal Structure of Rhodopsin: A G Protein-Coupled Receptor

3. Heterologous expression of G-protein-coupled receptors: comparison of expression systems from the standpoint of large-scale production and purification

4. Selective ligands as tools to study histamine receptors

Cited by 57 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Development of Conformationally Restricted Negamycin Derivatives for Potent Readthrough Activity;ACS Medicinal Chemistry Letters;2023-12-04

2. A stereochemical journey around spirocyclic glutamic acid analogs;Organic & Biomolecular Chemistry;2022

3. Modular Enantioselective Synthesis of cis-Cyclopropanes through Self-Sensitized Stereoselective Photodecarboxylation with Benzothiazolines;ACS Catalysis;2021-10-18

4. Enantioselective total synthesis of sesquiterpenoid phellilane L and its diastereomer;Tetrahedron;2021-05

5. Synthesis of Resolvin E1 and Its Conformationally Restricted Cyclopropane Congeners with Potent Anti-Inflammatory Effect;ACS Medicinal Chemistry Letters;2021-01-21