Automated Nanomole-Scale Reaction Screening toward Benzoate Bioisosteres: A Photocatalyzed Approach to Highly Elaborated Bicyclo[1.1.1]Pentanes-Reference-Cited by-同舟云学术

Automated Nanomole-Scale Reaction Screening toward Benzoate Bioisosteres: A Photocatalyzed Approach to Highly Elaborated Bicyclo[1.1.1]Pentanes

Published:2021-12-22 Issue:1 Volume:12 Page:600-606
ISSN:2155-5435
Container-title:ACS Catalysis
language:en
Short-container-title:ACS Catal.

Author:

Mousseau James J.¹^ORCID,Perry Matthew A.¹,Bundesmann Mark W.¹,Chinigo Gary M.¹,Choi Chulho¹^ORCID,Gallego Gary²^ORCID,Hicklin Robert W.¹,Hoy Susan¹,Limburg David C.¹,Sach Neal W.²,Zhang Yuan³^ORCID

Affiliation:

1. Pfizer Medicine Design, 445 Eastern Point Rd, Groton, Connecticut 06340, United States

2. Pfizer La Jolla Laboratories, 10770 Science Center Drive, San Diego, California 92121, United States

3. Pfizer Medicine Design, 610 Main St., Cambridge, Massachusetts 02139, United States

Publisher

American Chemical Society (ACS)

Subject

Catalysis,General Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acscatal.1c05076

Reference66 articles.

1. Escape from Flatland: Increasing Saturation as an Approach to Improving Clinical Success

2. Designing novel building blocks is an overlooked strategy to improve compound quality

3. The use of spirocyclic scaffolds in drug discovery

4. Two‐ and Three‐dimensional Rings in Drugs

5. 1-Substituted 2-Azaspiro[3.3]heptanes: Overlooked Motifs for Drug Discovery

Cited by 28 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Light-enabled scalable synthesis of bicyclo[1.1.1]pentane halides and their functionalizations;Nature Synthesis;2024-09-05

2. Photoinduced Multicomponent Heteroarylation of [1.1.1]Propellane with Katritzky Pyridinium Salts;Organic Letters;2024-08-14

3. Recent Advances in the Synthesis of Bicyclo[3.1.1]heptanes;Synthesis;2024-07-16

4. Addressing Reproducibility Challenges in High-Throughput Photochemistry;JACS Au;2024-06-27

5. A pharma perspective on sustainability advantages through adoption of continuous flow;Current Opinion in Green and Sustainable Chemistry;2024-04