Protein‐Templated Hit Identification through an Ugi Four‐Component Reaction**-Reference-Cited by-同舟云学术

Protein‐Templated Hit Identification through an Ugi Four‐Component Reaction**

Published:2020-09-30 Issue:64 Volume:26 Page:14585-14593
ISSN:0947-6539
Container-title:Chemistry – A European Journal
language:en
Short-container-title:Chem. Eur. J.

Author:

Mancini Federica¹²,Unver M. Yagiz¹³,Elgaher Walid A. M.¹^ORCID,Jumde Varsha R.¹,Alhayek Alaa¹²^ORCID,Lukat Peer⁴,Herrmann Jennifer⁵,Witte Martin D.³,Köck Matthias⁵,Blankenfeldt Wulf⁴⁶,Müller Rolf²⁵,Hirsch Anna K. H.¹²³^ORCID

Affiliation:

1. Department for Drug Design and Optimization Helmholtz Institute for Pharmaceutical Research Saarland (HIPS)–, Helmholtz Centre for Infection Research (HZI) Campus Building E8.1 66123 Saarbrücken Germany

2. Department of Pharmacy Saarland University Campus Building E8.1 66123 Saarbrücken Germany

3. Stratingh Institute for Chemistry University of Groningen Nijenborgh 7 9747 AG Groningen The Netherlands

4. Department of Structure and Function of Proteins HZI 38124 Braunschweig Germany

5. Department of Microbial Natural Products HIPS–HZI 66123 Saarbrücken Germany

6. Institute for Biochemistry, Biotechnology and Bioinformatics Technische Universität Braunschweig Spielmannstr. 7 38106 Braunschweig Germany

Publisher

Wiley

Subject

General Chemistry,Catalysis,Organic Chemistry

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/chem.202002250

Reference60 articles.

1. Protein-Templated Fragment Ligations-From Molecular Recognition to Drug Discovery

2. Proteintemplat-gesteuerte Fragmentligationen - von der molekularen Erkennung zur Wirkstofffindung

3. New insights into the kinetic target-guided synthesis of protein ligands

4. Druggability Assessment of Targets Used in Kinetic Target-Guided Synthesis

5. Kinetic Target-Guided Synthesis: Reaching the Age of Maturity

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