Selective Fragments for the CREBBP Bromodomain Identified from an Encoded Self‐assembly Chemical Library-Reference-Cited by-同舟云学术

Selective Fragments for the CREBBP Bromodomain Identified from an Encoded Self‐assembly Chemical Library

Published:2020-08-19 Issue:18 Volume:15 Page:1752-1756
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Catalano Marco¹,Moroglu Mustafa²,Balbi Petra¹,Mazzieri Federica¹,Clayton James²,Andrews Katrina H.²,Bigatti Martina³,Scheuermann Jörg¹,Conway Stuart J.²,Neri Dario¹^ORCID

Affiliation:

1. Department of Chemistry and Applied Biosciences Swiss Federal Institute of Technology (ETH Zürich) Vladimir-Prelog-Weg 4 8093 Zürich Switzerland

2. Department of Chemistry University of Oxford Mansfield Road Oxford OX1 3TA UK

3. Philochem AG 8112 Otelfingen Switzerland

Funder

Schweizerischer Nationalfonds zur Förderung der Wissenschaftlichen Forschung

Biotechnology and Biological Sciences Research Council

GlaxoSmithKline

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/cmdc.202000528

Reference30 articles.

1. Encoded combinatorial chemistry.

2. Reflections on DNA-encoded chemical libraries

3. DNA-encoded chemistry: enabling the deeper sampling of chemical space

4. Encoded Library Technologies as Integrated Lead Finding Platforms for Drug Discovery

5. Automated screening for small organic ligands using DNA-encoded chemical libraries

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