Discovery of novel 1,2,4‐triazole phenylalanine derivatives targeting an unexplored region within the interprotomer pocket of the HIV capsid protein-Reference-Cited by-同舟云学术

Discovery of novel 1,2,4‐triazole phenylalanine derivatives targeting an unexplored region within the interprotomer pocket of the HIV capsid protein

Published:2022-08-18 Issue:12 Volume:94 Page:5975-5986
ISSN:0146-6615
Container-title:Journal of Medical Virology
language:en
Short-container-title:Journal of Medical Virology

Author:

Jiang Xiangyi¹^ORCID,Sharma Prem Prakash²,Rathi Brijesh²,Ji Xiangkai¹,Hu Lide¹,Gao Zhen¹,Kang Dongwei¹³,Wang Zhao¹,Xie Minghui¹,Xu Shujing¹,Zhang Xujie¹,De Clercq Erik⁴,Cocklin Simon⁵,Pannecouque Christophe⁴,Dick Alexej⁵,Liu Xinyong¹³,Zhan Peng¹³

Affiliation:

1. Department of Medicinal Chemistry, Key Laboratory of Chemical Biology (Ministry of Education), School of Pharmaceutical Sciences, Cheeloo College of Medicine Shandong University Jinan Shandong China

2. Laboratory for Translational Chemistry and Drug Discovery, Department of Chemistry, Hansraj College University of Delhi Delhi India

3. China‐Belgium Collaborative Research Center for Innovative Antiviral Drugs of Shandong Province Shandong University Jinan Shandong China

4. Rega Institute for Medical Research, Laboratory of Virology and Chemotherapy K. U. Leuven Leuven Belgium

5. Department of Biochemistry & Molecular Biology Drexel University College of Medicine Philadelphia Pennsylvania USA

Publisher

Wiley

Subject

Infectious Diseases,Virology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/jmv.28064

Reference39 articles.

1. HIV-2 as a model to identify a functional HIV cure

2. Hiv-2 molecular epidemiology

3. In Vitro Antiviral Activity of Cabotegravir against HIV-2

4. Rapid initiation of antiretroviral therapy at HIV diagnosis: definition, process, knowledge gaps

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