A Series of Potent CREBBP Bromodomain Ligands Reveals an Induced-Fit Pocket Stabilized by a Cation-π Interaction-Reference-Cited by-同舟云学术

A Series of Potent CREBBP Bromodomain Ligands Reveals an Induced-Fit Pocket Stabilized by a Cation-π Interaction

Published:2014-05-12 Issue:24 Volume:126 Page:6240-6244
ISSN:0044-8249
Container-title:Angewandte Chemie
language:en
Short-container-title:Angew. Chem.

Author:

Rooney Timothy P. C.,Filippakopoulos Panagis,Fedorov Oleg,Picaud Sarah,Cortopassi Wilian A.,Hay Duncan A.,Martin Sarah,Tumber Anthony,Rogers Catherine M.,Philpott Martin,Wang Minghua,Thompson Amber L.,Heightman Tom D.,Pryde David C.,Cook Andrew,Paton Robert S.,Müller Susanne,Knapp Stefan,Brennan Paul E.,Conway Stuart J.

Publisher

Wiley

Subject

General Medicine

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