Synthesis and Opioid Activity of Tyr1-ψ[(Z)CF=CH]-Gly2and Tyr1-ψ[(S)/(R)-CF3CH-NH]-Gly2Leu-enkephalin Fluorinated Peptidomimetics-Reference-Cited by-同舟云学术

Synthesis and Opioid Activity of Tyr1-ψ[(Z)CF=CH]-Gly2and Tyr1-ψ[(S)/(R)-CF3CH-NH]-Gly2Leu-enkephalin Fluorinated Peptidomimetics

Published:2017-04-05 Issue:8 Volume:12 Page:571-576
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Karad Somnath Narayan¹,Pal Mohan¹,Crowley Rachel S.¹,Prisinzano Thomas E.¹^ORCID,Altman Ryan A.¹^ORCID

Affiliation:

1. Department of Medicinal Chemistry; The University of Kansas; 1251 Wescoe Hall Drive Lawrence Kansas 66045 USA

Funder

National Institute on Drug Abuse

National Institute of General Medical Sciences

National Institutes of Health

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Reference61 articles.

1. Opioid Abuse in Chronic Pain — Misconceptions and Mitigation Strategies

2. The Latest Prescription Trends for Controlled Prescription Drugs, 2015 www.drugabuse.gov/news-events/meetings-events/2015/09/latest-prescription-trends-controlled-prescription-drugs

3. Endogenous opiates and behavior: 2014

4. Trends in Drug-Poisoning Deaths Involving Opioid Analgesics and Heroin: United States, 1999-2012 2014 www.cdc.gov/nchs/data/hestat/drug_poisoning/drug_poisoning.htm

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