Fragments as Novel Starting Points for tRNA‐Guanine Transglycosylase Inhibitors Found by Alternative Screening Strategies-Reference-Cited by-同舟云学术

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Fragments as Novel Starting Points for tRNA‐Guanine Transglycosylase Inhibitors Found by Alternative Screening Strategies

Published:2020-01-29 Issue:3 Volume:15 Page:324-337
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Hassaan Engi¹^ORCID,Eriksson Per‐Olof²^ORCID,Geschwindner Stefan²^ORCID,Heine Andreas¹^ORCID,Klebe Gerhard¹^ORCID

Affiliation:

1. Institute of Pharmaceutical Chemistry Philipps University Marburg Marbacher Weg 6 35032 Marburg Germany

2. Structure, Biophysics and Fragment-based Lead Generation Discovery Sciences, R&D, AstraZeneca 431 83 Gothenburg Sweden

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/cmdc.201900604

Reference46 articles.

1. Fragment-Based Lead Discovery and Design

2. F. U. Huschmann J. Linnik K. Sparta M. Uehlein X. Wang A. Metz J. Schiebel A. Heine G. Klebe M. S. Weiss U. Mueller Acta Crystallogr. Sect. F: Struct. Biol. Commun.2016 72 346–355.

3. https://www.jenabioscience.com/crystallography-cryo-em/screening/fragment-screen.

4. A ‘Rule of Three’ for fragment-based lead discovery?

5. A Small Nonrule of 3 Compatible Fragment Library Provides High Hit Rate of Endothiapepsin Crystal Structures with Various Fragment Chemotypes

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