Synthesis of All‐Carbon Disubstituted Bicyclo[1.1.1]pentanes by Iron‐Catalyzed Kumada Cross‐Coupling-Reference-Cited by-同舟云学术

Synthesis of All‐Carbon Disubstituted Bicyclo[1.1.1]pentanes by Iron‐Catalyzed Kumada Cross‐Coupling

Published:2020-05-14 Issue:29 Volume:132 Page:11964-11968
ISSN:0044-8249
Container-title:Angewandte Chemie
language:en
Short-container-title:Angew. Chem.

Author:

Nugent Jeremy¹^ORCID,Shire Bethany R.¹,Caputo Dimitri F. J.¹^ORCID,Pickford Helena D.¹,Nightingale Frank¹,Houlsby Ian T. T.²,Mousseau James J.³^ORCID,Anderson Edward A.¹^ORCID

Affiliation:

1. Chemistry Research Laboratory University of Oxford 12 Mansfield Road Oxford OX1 3TA UK

2. Syngenta Ltd. Jealott's Hill International Research Centre Bracknell RG42 6EY UK

3. Pfizer Medicine Design Eastern Point Road Groton CT 06340 USA

Funder

Engineering and Physical Sciences Research Council

H2020 Marie Skłodowska-Curie Actions

Royal Society of Chemistry

Publisher

Wiley

Subject

General Medicine

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/ange.202004090

Reference79 articles.

2. Improving Nonspecific Binding and Solubility: Bicycloalkyl Groups and Cubanes as para -Phenyl Bioisosteres

3. Application of the Bicyclo[1.1.1]pentane Motif as a Nonclassical Phenyl Ring Bioisostere in the Design of a Potent and Orally Active γ-Secretase Inhibitor

4. Investigation of a Bicyclo[1.1.1]pentane as a Phenyl Replacement within an LpPLA2 Inhibitor

5. Toward Resolving the Resveratrol Conundrum: Synthesis and in Vivo Pharmacokinetic Evaluation of BCP–Resveratrol

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