Design and synthesis of 1,2,4‐triazolo[1,5‐a]pyrimidine derivatives as PDE 4B inhibitors endowed with bronchodilator activity-Reference-Cited by-同舟云学术

Design and synthesis of 1,2,4‐triazolo[1,5‐a]pyrimidine derivatives as PDE 4B inhibitors endowed with bronchodilator activity

Published:2019-07-29 Issue:8 Volume:352 Page:1900002
ISSN:0365-6233
Container-title:Archiv der Pharmazie
language:en
Short-container-title:Arch Pharm Chem Life Sci

Author:

Abd El‐Aleam Rehab H.¹,George Riham F.²^ORCID,Lee Kevin J.³,Keeton Adam B.³,Piazza Gary A.³,Kamel Amr A.⁴,El‐Daly Mahmoud E.⁴,Hassan Ghaneya S.²⁵,Abdel‐Rahman Hamdy M.¹⁶

Affiliation:

1. Pharmaceutical Chemistry Department, Faculty of PharmacyNahda University Beni Suef Egypt

2. Pharmaceutical Chemistry Department, Faculty of PharmacyCairo University Cairo Egypt

3. USA Mitchell Cancer Institute Drug Discovery LaboratoryUniversity of South Alabama Mobile Alabama

4. Pharmacology and Toxicology Department, Faculty of PharmacyMinia University El‐Minia Egypt

5. Pharmaceutical Chemistry Department, Faculty of PharmacyBadr University Badr City Cairo Egypt

6. Medicinal Chemistry Department, Faculty of PharmacyAssiut University Assiut Egypt

Publisher

Wiley

Subject

Drug Discovery,Pharmaceutical Science

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/ardp.201900002

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4. Recent Advances on Phosphodiesterase 4 Inhibitors for the Treatment of Asthma and Chronic Obstructive Pulmonary Disease

5. PDE4D promotes FAK-mediated cell invasion in BRAF-mutated melanoma

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