High-throughput cytochrome P450 (CYP) inhibition screening via a cassette probe-dosing strategy. VI. Simultaneous evaluation of inhibition potential of drugs on human hepatic isozymes CYP2A6, 3A4, 2C9, 2D6 and 2E1-Reference-Cited by-同舟云学术

High-throughput cytochrome P450 (CYP) inhibition screening via a cassette probe-dosing strategy. VI. Simultaneous evaluation of inhibition potential of drugs on human hepatic isozymes CYP2A6, 3A4, 2C9, 2D6 and 2E1

Published:2001 Issue:10 Volume:15 Page:741-748
ISSN:0951-4198
Container-title:Rapid Communications in Mass Spectrometry
language:en
Short-container-title:Rapid Commun. Mass Spectrom.

Author:

Bu Hai-Zhi,Magis Lisa,Knuth Kim,Teitelbaum Philip

Publisher

Wiley

Subject

Organic Chemistry,Spectroscopy,Analytical Chemistry

Reference19 articles.

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2. Inhibitors of P450-dependent steroid biosynthesis: From research to medical treatment

3. Automated high throughput human CYP isoform activity assay using SPE-LC/MS method: application in CYP inhibition evaluation

4. Fully automated analysis of activities catalysed by the major human liver cytochrome P450 (CYP) enzymes: assessment of human CYP inhibition potential

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