Bisubstrate Inhibitors of CatecholO-Methyltransferase (COMT): the Crucial Role of the Ribose Structural Unit for Inhibitor Binding Affinity-Reference-Cited by-同舟云学术

Bisubstrate Inhibitors of CatecholO-Methyltransferase (COMT): the Crucial Role of the Ribose Structural Unit for Inhibitor Binding Affinity

Published:2006-03-13 Issue:3 Volume:1 Page:340-357
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Paulini Ralph,Trindler Christian,Lerner Christian,Brändli Lukas,Schweizer W. Bernd,Jakob-Roetne Roland,Zürcher Gerhard,Borroni Edilio,Diederich François

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Reference85 articles.

1. Kinetic inhibitory profile of BIA 3-202, a novel fast tight-binding, reversible and competitive catechol-O-methyltransferase inhibitor

2. COMT Inhibition in the Treatment of Parkinson’S Disease: Neuroprotection and Future Perspectives

3. Prefrontal neurons and the genetics of schizophrenia

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