Author:
Heinrich Timo,Böttcher Henning,Prücher Helmut,Gottschlich Rudolf,Ackermann Karl-August,van Amsterdam Christoph
Subject
Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology
Cited by
12 articles.
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1. Development of novel conformationally restricted selective Clk1/4 inhibitors through creating an intramolecular hydrogen bond involving an imide linker;European Journal of Medicinal Chemistry;2022-08
2. Synthesis of 2,3-dihydrobenzo[b][1,4]dioxine-5-carboxamide and 3-oxo-3,4-dihydrobenzo[b][1,4]oxazine-8-carboxamide derivatives as PARP1 inhibitors;Bioorganic Chemistry;2020-09
3. Design, Synthesis, and Pharmacological Characterization of Heterobivalent Ligands for the Putative 5-HT2A/mGlu2 Receptor Complex;Journal of Medicinal Chemistry;2020-08-20
4. Targeting Serotonin 2A and Adrenergic α
1
Receptors for Ocular Antihypertensive Agents: Discovery of 3,4‐Dihydropyrazino[1,2‐
b
]indazol‐1(2
H
)‐one Derivatives;ChemMedChem;2018-07-09
5. Molecular pharmacophore selectivity studies, virtual screening, and in silico ADMET analysis of GPCR antagonists;Medicinal Chemistry Research;2015-07-14