Synthesis of 2,3-dihydrobenzo[b][1,4]dioxine-5-carboxamide and 3-oxo-3,4-dihydrobenzo[b][1,4]oxazine-8-carboxamide derivatives as PARP1 inhibitors-Reference-Cited by-同舟云学术

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Synthesis of 2,3-dihydrobenzo[b][1,4]dioxine-5-carboxamide and 3-oxo-3,4-dihydrobenzo[b][1,4]oxazine-8-carboxamide derivatives as PARP1 inhibitors

Published:2020-09 Issue: Volume:102 Page:104075
ISSN:0045-2068
Container-title:Bioorganic Chemistry
language:en
Short-container-title:Bioorganic Chemistry

Author:

Shao Xuwei,Pak Steven,Velagapudi Uday Kiran,Gobbooru Shruthi,Kommaraju Sai Shilpa,Low Woon-Kai,Subramaniam Gopal,Pathak Sanjai Kumar,Talele Tanaji T.

Funder

Department of Pharmaceutical Sciences of St. John’s University

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

Reference28 articles.

1. PARP-1 mechanism for coupling DNA damage detection to poly(ADP-ribose) synthesis;Langelier;Curr. Opin. Struct. Biol.,2013

2. A phase I study of topotecan, carboplatin and the PARP inhibitor veliparib in acute leukemias, aggressive myeloproliferative neoplasms, and chronic myelomonocytic leukemia;Pratz;Clin. Cancer Res.,2017

3. A phase I clinical trial of the poly(ADP-ribose) polymerase inhibitor veliparib and weekly topotecan in patients with solid tumors;Wahner Hendrickson;Clin. Cancer Res.,2018

4. Specific killing of BRCA2-deficient tumours with inhibitors of poly(ADP-ribose) polymerase;Bryant;Nature,2005

5. Targeting the DNA repair defect in BRCA mutant cells as a therapeutic strategy;Farmer;Nature,2005

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1. The recent advance and prospect of poly(ADP‐ribose) polymerase inhibitors for the treatment of cancer;Medicinal Research Reviews;2024-08-24

2. Targeting selective inhibitors of PARPs in drug discovery and development;Medicinal Chemistry Research;2024-07-28

3. Synthetic PARP-1 Inhibitors Reported During the Last Decade;Letters in Drug Design & Discovery;2023-07

4. Ring-Opening Cyclization (ROC) of Aziridines with Propargyl Alcohols: Synthesis of 3,4-Dihydro-2H-1,4-oxazines;The Journal of Organic Chemistry;2023-03-27

5. Selective PARP1 inhibitors, PARP1-based dual-target inhibitors, PROTAC PARP1 degraders, and prodrugs of PARP1 inhibitors for cancer therapy;Pharmacological Research;2022-12

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