Activity and selectivity cliffs for DPP-IV inhibitors: Lessons we can learn from SAR studies and their application to virtual screening
Author:
Affiliation:
1. Research Group in Cheminformatics & Nutrition, Departament de Bioquímica i Biotecnologia; Universitat Rovira i Virgili; Campus de Sescelades; Tarragona Spain
2. EURECAT, TECNIO, CEICS; Avinguda Universitat 1; Reus Spain
Funder
Agència de Gestió d’Ajuts Universitaris i de Recerca
Programa de Foment de la Recerca (URV)
Publisher
Wiley
Subject
Drug Discovery,Pharmacology,Molecular Medicine
Link
http://onlinelibrary.wiley.com/wol1/doi/10.1002/med.21499/fullpdf
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3. Dipeptidyl-peptidase 4 inhibition: linking metabolic control to cardiovascular protection;Avogaro;Curr Pharm Des,2013
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