Implications of Dynamic Occupancy, Binding Kinetics, and Channel Gating Kinetics for hERG Blocker Safety Assessment and Mitigation-Reference-Cited by-同舟云学术

Implications of Dynamic Occupancy, Binding Kinetics, and Channel Gating Kinetics for hERG Blocker Safety Assessment and Mitigation

Published:2016-04-29 Issue:16 Volume:16 Page:1792-1818
ISSN:1568-0266
Container-title:Current Topics in Medicinal Chemistry
language:en
Short-container-title:CTMC

Author:

A. Pearlstein Robert,Andrew MacCannell K.,Erdemli Gül,Yeola Sarita,Helmlinger Gabriel,Hu Qi-Ying,Farid Ramy,Egan William,Whitebread Steven,Springer Clayton,Beck Jeremy,Wang Hao-Ran,Maciejewski Mateusz,Urban Laszlo,S. Duca José

Publisher

Bentham Science Publishers Ltd.

Subject

Drug Discovery,General Medicine

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