Aromatase: The Enzyme and Its Inhibition-Reference-Cited by-同舟云学术

Aromatase: The Enzyme and Its Inhibition

Published:2009-07-01 Issue:6 Volume:9 Page:627-641
ISSN:1871-5206
Container-title:Anti-Cancer Agents in Medicinal Chemistry
language:en
Short-container-title:ACAMC

Author:

Banting Lee,Ahmed Sabbir¹

Affiliation:

1. School of Pharmacy and Biomedical Sciences, University of Portsmouth, St. Michael's Building, White Swan Road, Portsmouth PO1 2DT, UK.

Abstract

The genetic control, mechanism of action and inhibition of aromatase for potential therapeutic benefits in the arena of hormone dependent illness continues to be of considerable interest. The work presented here concentrates on recent advances in the mechanistic aspects of the aromatase enzyme and the nature of the chemical entities that lead to its inhibition.

Publisher

Bentham Science Publishers Ltd.

Subject

Cancer Research,Pharmacology,Molecular Medicine

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1. Working at the membrane interface: Ligand-induced changes in dynamic conformation and oligomeric structure in human aromatase;Biotechnology and Applied Biochemistry;2017-10-23

2. Computational insights into inhibitory mechanism of azole compounds against human aromatase;RSC Advances;2015

3. Computational Approaches Elucidate the Allosteric Mechanism of Human Aromatase Inhibition: A Novel Possible Route to Small-Molecule Regulation of CYP450s Activities?;Journal of Chemical Information and Modeling;2014-09-15

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