Bridging the gap: bitopic ligands of G-protein-coupled receptors
Author:
Publisher
Elsevier BV
Subject
Pharmacology,Toxicology
Reference55 articles.
1. Progress in structure based drug design for G protein-coupled receptors;Congreve;J. Med. Chem.,2011
2. Structural diversity of G protein-coupled receptors and significance for drug discovery;Lagerström;Nat. Rev. Drug Discov.,2008
3. Seven transmembrane receptors as shapeshifting proteins: the impact of allosteric modulation and functional selectivity on new drug discovery;Kenakin;Pharmacol. Rev.,2010
4. Allosteric GPCR modulators: taking advantage of permissive receptor pharmacology;Leach;Trends Pharmacol. Sci.,2007
5. Allosteric modulation of G protein-coupled receptors;May;Annu. Rev. Pharmacol. Toxicol.,2007
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