Pharmacological and antihyperalgesic properties of the novel α2/3 preferring GABA A receptor ligand MP-III-024-Reference-Cited by-同舟云学术

Pharmacological and antihyperalgesic properties of the novel α2/3 preferring GABA A receptor ligand MP-III-024

Published:2017-05 Issue: Volume:131 Page:62-69
ISSN:0361-9230
Container-title:Brain Research Bulletin
language:en
Short-container-title:Brain Research Bulletin

Author:

Fischer Bradford D.,Schlitt Raymond J.,Hamade Bryan Z.,Rehman Sabah,Ernst Margot,Poe Michael M.,Li Guanguan,Kodali Revathi,Arnold Leggy A.,Cook James M.

Publisher

Elsevier BV

Subject

General Neuroscience

Reference41 articles.

1. GABAA receptor subtype-selective modulators. II. α5-selective inverse agonists for cognition enhancement;Atack;Curr. Top. Med. Chem.,2011

2. Enhanced learning and memory and altered GABAergic synaptic transmission in mice lacking the alpha 5 subunit of the GABAA receptor;Collinson;J. Neurosci.,2002

3. Trace fear conditioning involves hippocampal alpha5 GABA(A) receptors;Crestani;Proc. Natl. Acad. Sci. U. S. A.,2002

4. GABAA α5 subunit-containing receptors do not contribute to reversal of inflammatory-induced spinal sensitization as indicated by the unique selectivity profile of the GABAA receptor allosteric modulator NS16085;de Lucas;Biochem. Pharmacol.,2015

5. HZ166, a novel GABAA receptor subtype-selective benzodiazepine site ligand, is antihyperalgesic in mouse models of inflammatory and neuropathic pain;Di Lio;Neuropharmacology,2011

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