When simple agonism is not enough: Emerging modalities of GPCR ligands-Reference-Cited by-同舟云学术

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When simple agonism is not enough: Emerging modalities of GPCR ligands

Published:2011-01 Issue:2 Volume:331 Page:241-247
ISSN:0303-7207
Container-title:Molecular and Cellular Endocrinology
language:en
Short-container-title:Molecular and Cellular Endocrinology

Author:

Smith Nicola J.,Bennett Kirstie A.,Milligan Graeme

Funder

Biotechnology and Biological Sciences Research Council (BBSRC)

Publisher

Elsevier BV

Subject

Endocrinology,Molecular Biology,Biochemistry

Reference87 articles.

1. Dualsteric GPCR targeting: a novel route to binding and signaling pathway selectivity;Antony;FASEB J.,2009

2. Growth hormone secretagogues and growth hormone releasing peptides act as orthosteric super-agonists but not allosteric regulators for activation of the G protein Galpha(o1) by the Ghrelin receptor;Bennett;Mol. Pharmacol.,2009

3. A bivalent ligand (KDN-21) reveals spinal delta and kappa opioid receptors are organized as heterodimers that give rise to delta(1) and kappa(2) phenotypes. Selective targeting of delta-kappa heterodimers;Bhushan;J. Med. Chem.,2004

4. The heptahelical domain of GABA(B2) is activated directly by CGP7930, a positive allosteric modulator of the GABA(B) receptor;Binet;J. Biol. Chem.,2004

5. Allosterism at muscarinic receptors: ligands and mechanisms;Birdsall;Mini Rev. Med. Chem.,2005

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