Synthesis and Structure–Activity relationship of 1-(5-isoquinolinesulfonyl)piperazine analogues as inhibitors of Mycobacterium tuberculosis IMPDH-Reference-Cited by-同舟云学术

Synthesis and Structure–Activity relationship of 1-(5-isoquinolinesulfonyl)piperazine analogues as inhibitors of Mycobacterium tuberculosis IMPDH

Published:2019-07 Issue: Volume:174 Page:309-329
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Singh Vinayak^ORCID,Pacitto Angela,Donini Stefano,Ferraris Davide M.,Boros Sándor,Illyés Eszter,Szokol Bálint^ORCID,Rizzi Menico,Blundell Tom L.,Ascher David B.,Pato Janos,Mizrahi Valerie

Funder

European Community’s Seventh Framework Programme

Howard Hughes Medical Institute

National Research Foundation of South Africa

South African Medical Research Council

Jack Brockhoff Foundation

National Health and Medical Research Council of Australia

Department of Biochemistry, University of Melbourne

Newton Fund RCUK-CONFAP

Medical Research Council

Fundação de Amparo à Pesquisa do Estado de Minas Gerais

Bill and Melinda Gates Foundation

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

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