The Inosine Monophosphate Dehydrogenase, GuaB2, Is a Vulnerable New Bactericidal Drug Target for Tuberculosis

Author:

Singh Vinayak1,Donini Stefano2,Pacitto Angela3,Sala Claudia4,Hartkoorn Ruben C.4,Dhar Neeraj4,Keri Gyorgy5,Ascher David B.3,Mondésert Guillaume6,Vocat Anthony4,Lupien Andréanne4,Sommer Raphael4,Vermet Hélène6,Lagrange Sophie6,Buechler Joe7,Warner Digby F.1,McKinney John D.4,Pato Janos5,Cole Stewart T.4,Blundell Tom L.3,Rizzi Menico2,Mizrahi Valerie1

Affiliation:

1. MRC/NHLS/UCT Molecular Mycobacteriology Research Unit & DST/NRF Centre of Excellence for Biomedical TB Research, Institute of Infectious Disease and Molecular Medicine & Department of Pathology, University of Cape Town, Anzio Road, Observatory 7925, South Africa

2. Dipartimento di Scienze del Farmaco, University of Piemonte Orientale, Via Bovio 6, 28100 Novara, Italy

3. Department of Biochemistry, University of Cambridge, 80 Tennis Court Road, Cambridge CB2 1GA, United Kingdom

4. Ecole Polytechnique Fédérale de Lausanne, Global Health Institute, Station 19, 1015 Lausanne, Switzerland

5. Vichem Chemie, Herman Ottó út 15, Budapest, 1022 Hungary

6. Sanofi-Aventis Research & Development, Infectious Diseases Unit, Biology Group, Campus Mérieux, 1541 avenue Marcel Mérieux, 69280 Marcy L’Etoile, France

7. Alere (San Diego), Summer Ridge Road, San Diego, California 92121, United States

Funder

Howard Hughes Medical Institute

Fundação de Amparo à Pesquisa do Estado de Minas Gerais

National Health and Medical Research Council

Bill and Melinda Gates Foundation

National Research Foundation

Seventh Framework Programme

South African Medical Research Council

Fondation Jacqueline Beytout

Swiss National Science Foundation

Publisher

American Chemical Society (ACS)

Subject

Infectious Diseases

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