Novel 2-(2-arylmethylthio-4-chloro-5-methylbenzenesulfonyl)-1-(1,3,5-triazin-2-ylamino)guanidine derivatives: Inhibition of human carbonic anhydrase cytosolic isozymes I and II and the transmembrane tumor-associated isozymes IX and XII, anticancer activity, and molecular modeling studies-Reference-Cited by-同舟云学术

Novel 2-(2-arylmethylthio-4-chloro-5-methylbenzenesulfonyl)-1-(1,3,5-triazin-2-ylamino)guanidine derivatives: Inhibition of human carbonic anhydrase cytosolic isozymes I and II and the transmembrane tumor-associated isozymes IX and XII, anticancer activity, and molecular modeling studies

Published:2018-01 Issue: Volume:143 Page:1931-1941
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Żołnowska Beata,Sławiński Jarosław,Szafrański Krzysztof,Angeli Andrea,Supuran Claudiu T.,Kawiak Anna,Wieczór Miłosz^ORCID,Zielińska Joanna,Bączek Tomasz,Bartoszewska Sylwia

Funder

PL-Grid infrastructure

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference47 articles.

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3. Carbonic anhydrases: novel therapeutic applications for inhibitors and activators;Supuran;Nat. Rev. Drug Discov.,2008

4. Amido/ureidosubstituted benzenesulfonamides-isatin conjugates as low nanomolar/subnanomolar inhibitors of the tumor-associated carbonic anhydrase isoform XII;Eldehna;Eur. J. Med. Chem.,2016

5. Synthesis, carbonic anhydrase inhibition and cytotoxic activity of novel chromone-based sulfonamide derivatives;Awadallah;Eur. J. Med. Chem.,2015

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