Discovery of potent IDO1 inhibitors derived from tryptophan using scaffold-hopping and structure-based design approaches-Reference-Cited by-同舟云学术

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Discovery of potent IDO1 inhibitors derived from tryptophan using scaffold-hopping and structure-based design approaches

Published:2017-09 Issue: Volume:138 Page:199-211
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Zou Yi^ORCID,Wang Yan,Wang Fang,Luo Minghao,Li Yuezhen,Liu Wen,Huang Zhangjian,Zhang Yihua,Guo Wenjie,Xu Qiang,Lai Yisheng

Funder

National Natural Science Foundation of China

Jiangsu Province Funds for Distinguished Young Scientists

Six Major Talent Peak Project of Jiangsu Province

Fundamental Research Funds for the Central Universities

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference55 articles.

1. Immune evasion in cancer: mechanistic basis and therapeutic strategies;Vinay;Semin. Cancer Biol.,2015

2. IDO in the tumor microenvironment: inflammation, counter-regulation, and tolerance;Munn;Trends Immunol.,2016

3. Tryptophan catabolism in cancer: beyond IDO and tryptophan depletion;Platten;Cancer Res.,2012

4. Extensive profiling of the expression of the indoleamine 2,3-dioxygenase 1 protein in normal and tumoral human tissues;Théate;Cancer Immunol. Res.,2015

5. Constitutive IDO expression in human cancer is sustained by an autocrine signaling loop involving IL-6, STAT3 and the AHR;Litzenburger;Oncotarget,2014

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