4-Hydroxy-1,2,3-triazole moiety as bioisostere of the carboxylic acid function: a novel scaffold to probe the orthosteric γ-aminobutyric acid receptor binding site-Reference-Cited by-同舟云学术

4-Hydroxy-1,2,3-triazole moiety as bioisostere of the carboxylic acid function: a novel scaffold to probe the orthosteric γ-aminobutyric acid receptor binding site

Published:2018-10 Issue: Volume:158 Page:311-321
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Giraudo Alessandro^ORCID,Krall Jacob,Nielsen Birgitte,Sørensen Troels E.,Kongstad Kenneth T.,Rolando Barbara^ORCID,Boschi Donatella^ORCID,Frølund Bente,Lolli Marco L.^ORCID

Funder

University of Turin

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference52 articles.

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5. Novel 4-(piperidin-4-yl)-1-hydroxypyrazoles as gamma-aminobutyric acid(A) receptor ligands: synthesis, pharmacology, and structure-activity relationships;Moller;J. Med. Chem.,2010

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