Exploring the role of the 5′-position of TSAO-T. Synthesis and anti-HIV evaluation of novel TSAO-T derivatives
Author:
Publisher
Elsevier BV
Subject
Virology,Pharmacology
Reference33 articles.
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4. 2′,5′-Bis-O-(tert-butyldimethylsilyl)-3′-spiro-5″-(4″-amino-1″,2″-oxathiole-2″,2″-dioxide) pyrimidine (TSAO) nucleoside analogues: highly selective inhibitors of human immunodeficiency virus type 1 that are targeted at the viral reverse transcriptase;Balzarini;Proc. Natl. Acad. Sci. USA,1992
5. 2′,5′-Bis-O-(tert-butyldimethylsilyl)]-3′-spiro-5″-(4″-amino-1″,2″-oxathiole-2″,2″-dioxide) (TSAO) derivatives of purine and pyrimidine nucleosides as potent and selective inhibitors of human immunodeficiency virus type 1;Balzarini;Antimicrob. Agents Chemother.,1992
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