Design and synthesis of novel protease inhibitors. Tripeptide α′,β′-epoxyketones as nanomolar inactivators of the proteasome-Reference-Cited by-同舟云学术

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Design and synthesis of novel protease inhibitors. Tripeptide α′,β′-epoxyketones as nanomolar inactivators of the proteasome

Published:1996-02 Issue:9 Volume:37 Page:1343-1346
ISSN:0040-4039
Container-title:Tetrahedron Letters
language:en
Short-container-title:Tetrahedron Letters

Author:

Spaltenstein Andrew,Leban Johann J.,Huang Jim J.,Reinhardt Kelli R.,Humberto Viveros O.,Sigafoos Jim,Crouch Ronald

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Reference18 articles.

1. Crystal Structure of the 20 S Proteasome from the Archaeon T. acidophilum at 3.4 Å Resolution

2. Proteasome from Thermoplasma acidophilum : a Threonine Protease

3. The ubiquitinproteasome pathway is required for processing the NF-κB1 precursor protein and the activation of NF-κB

4. Ubiquitin-dependent c-Jun degradation in vivo is mediated by the δ domain

5. The E6 oncoprotein encoded by human papillomavirus types 16 and 18 promotes the degradation of p53

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1. Natural product scaffolds as inspiration for the design and synthesis of 20S human proteasome inhibitors;RSC Chemical Biology;2020

2. Binding of the Microbial Cyclic Tetrapeptide Trapoxin A to the Class I Histone Deacetylase HDAC8;ACS Chemical Biology;2017-08-30

3. A new strategy for accessing (S)-1-(furan-2-yl)pent-4-en-1-ol: a key precursor of Ipomoeassin family of compounds and C1–C15 domain of halichondrins;Tetrahedron Letters;2016-08

4. Total synthesis of isocladosporin and 3- epi -isocladosporin;Tetrahedron Letters;2016-01

5. Design, Synthesis and Biological Evaluation of Peptidyl Epoxyketone Proteasome Inhibitors Composed ofβ-amino Acids;Chemical Biology & Drug Design;2014-06-03

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