Development of potent dimeric inhibitors of GAS41 YEATS domain-Reference-Cited by-同舟云学术

Development of potent dimeric inhibitors of GAS41 YEATS domain

Published:2021-12 Issue:12 Volume:28 Page:1716-1727.e6
ISSN:2451-9456
Container-title:Cell Chemical Biology
language:en
Short-container-title:Cell Chemical Biology

Author:

Listunov Dymytrii^ORCID,Linhares Brian M.^ORCID,Kim EunGi^ORCID,Winkler Alyssa,Simes Miranda L.^ORCID,Weaver Sidney^ORCID,Cho Hyo Je^ORCID,Rizo Alexandrea^ORCID,Zolov Sergey,Keshamouni Venkateshwar G.,Grembecka Jolanta,Cierpicki Tomasz

Publisher

Elsevier BV

Subject

Clinical Biochemistry,Drug Discovery,Pharmacology,Molecular Biology,Molecular Medicine,Biochemistry

Reference37 articles.

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3. The Taf14 YEATS domain is a reader of histone crotonylation;Andrews;Nat. Chem. Biol.,2016

4. Subtype-specific genomic alterations define new targets for soft-tissue sarcoma therapy;Barretina;Nat. Genet.,2010

5. GAS41 recognizes diacetylated histone H3 through a bivalent binding mode;Cho;ACS Chem. Biol.,2018

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1. YEATS domain-containing protein GAS41 regulates nuclear shape by working in concert with BRD2 and the mediator complex in colorectal cancer;Pharmacological Research;2024-08

2. Therapeutic targeting of BET bromodomain and other epigenetic acetylrecognition domain–containing factors;Current Opinion in Genetics & Development;2024-06

3. GAS41 modulates ferroptosis by anchoring NRF2 on chromatin;Nature Communications;2024-03-21

4. Discovery of PFI-6, a small-molecule chemical probe for the YEATS domain of MLLT1 and MLLT3;Bioorganic & Medicinal Chemistry Letters;2024-01

5. Small-molecule tools for YEATS domain proteins;Current Opinion in Chemical Biology;2023-12