Discovery of PFI-6, a small-molecule chemical probe for the YEATS domain of MLLT1 and MLLT3-Reference-Cited by-同舟云学术

Discovery of PFI-6, a small-molecule chemical probe for the YEATS domain of MLLT1 and MLLT3

Published:2024-01 Issue: Volume:98 Page:129546
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Raux Brigitt,Buchan Karly A.,Bennett James,Christott Thomas,Dowling Matthew S.,Farnie Gillian,Fedorov Oleg,Gamble Vicki,Gileadi Carina,Giroud Charline^ORCID,Huber Kilian V.M.^ORCID,Korczynska Magdalena,Limberakis Chris^ORCID,Narayanan Arjun,Owen Dafydd R.,Sáez Laura Díaz^ORCID,Stock Ingrid A.,Londregan Allyn T.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference45 articles.

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2. Patel, D. J. How chromatin-binding modules interpret histone modifications. Nat Struct Mol Biol. 2007, 14, 1025-1040. (c) Musselman, C. A.

3. Kutateladze, T. G. Perceiving the epigenetic landscape through histone readers. Nat Struct Mol Biol. 2012, 19, 1218-1227.

4. (a) Strahl, B. D.; Allis, C. D. The language of covalent histone modifications. Nature. 2000, 40, 41-45.

5. (b) Taverna, S. D.; Li, H.; Ruthenburg, A. J., Allis, C. D.; Patel, D. J. How chromatin-binding modules interpret histone modifications. Nat Struct Mol Biol. 2007, 14, 1025-1040.

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