Synthesis and initial in vitro characterization of a new P2X7R radioligand [18F]IUR-1602-Reference-Cited by-同舟云学术

Synthesis and initial in vitro characterization of a new P2X7R radioligand [18F]IUR-1602

Published:2019-02 Issue: Volume:144 Page:10-18
ISSN:0969-8043
Container-title:Applied Radiation and Isotopes
language:en
Short-container-title:Applied Radiation and Isotopes

Author:

Gao Mingzhang,Wang Min,Glick-Wilson Barbara E.,Meyer Jill A.,Peters Jonathan S.,Territo Paul R.,Green Mark A.,Hutchins Gary D.,Zarrinmayeh Hamideh,Zheng Qi-Huang

Funder

Indiana University Showalter Young Investigator Award

Indiana University Department of Radiology and Imaging Sciences

National Science Foundation

Publisher

Elsevier BV

Subject

Radiation

Reference26 articles.

1. SPECT imaging of dopamine transporters in human brain with iodine-123-fluoroalkyl analogs of β-CIT;Abi-Dargham;J. Nucl. Med.,1996

2. Design, synthesis and evaluation in an LPS rodent model of neuroinflammation of a novel 18F-labelled PET tracer targeting P2X7;Fantoni;EJNMMI Res.,2017

3. Synthesis and preliminary biological evaluation of a novel P2X7R radioligand [18F]IUR-1601;Gao;Bioorg. Med. Chem. Lett.,2018

4. Synthesis of [11C]GSK1482160 as a new PET agent for targeting P2X7 receptor;Gao;Bioorg. Med. Chem. Lett.,2015

5. Synthesis and preliminary biological evaluation of [11C]methyl (2-amino-5-(benzylthio)thiazolo[4,5-d]pyrimidin-7-yl)-d-leucinate for the fractalkine receptor (CX3CR1);Gao;Bioorg. Med. Chem. Lett.,2017

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