Orally bioavailable, indole-based nonpeptide GnRH receptor antagonists with high potency and functional activity-Reference-Cited by-同舟云学术

Orally bioavailable, indole-based nonpeptide GnRH receptor antagonists with high potency and functional activity

Published:2001-10 Issue:19 Volume:11 Page:2597-2602
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Ashton Wallace T.,Sisco Rosemary M.,Kieczykowski Gerard R.,Yang Yi Tien,Yudkovitz Joel B.,Cui Jisong,Mount George R.,Ren Rena Ning,Wu Tsuei-Ju,Shen Xiaolan,Lyons Kathryn A.,Mao An-Hua,Carlin Josephine R.,Karanam Bindhu V.,Vincent Stella H.,Cheng Kang,Goulet Mark T.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference29 articles.

1. Progress towards the development of non-peptide orally-active gonadotropin-releasing hormone (GnRH) antagonists: therapeutic implications

2. Discovery of a Novel, Potent, and Orally Active Nonpeptide Antagonist of the Human Luteinizing Hormone-Releasing Hormone (LHRH) Receptor

3. Chemistry and Molecular Biology in the Search for New LHRH Antagonists

4. Initial structure–activity relationship of a novel class of nonpeptidyl GnRH receptor antagonists: 2-arylindoles

5. SAR studies of novel 5-substituted 2-arylindoles as nonpeptidyl GnRH receptor antagonists

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