Discovery of thienopyrimidine-based inhibitors of the human farnesyl pyrophosphate synthase—Parallel synthesis of analogs via a trimethylsilyl ylidene intermediate-Reference-Cited by-同舟云学术

Discovery of thienopyrimidine-based inhibitors of the human farnesyl pyrophosphate synthase—Parallel synthesis of analogs via a trimethylsilyl ylidene intermediate

Published:2013-04 Issue:8 Volume:21 Page:2229-2240
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Leung Chun-Yuen,Langille Adrienne M.,Mancuso John,Tsantrizos Youla S.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference40 articles.

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3. Brewster, W. K.; Klittich, C. J. R.; Balko, T.W.; Breax, N. T.; Erickson, W. R.; Hunter, J. E.; Lowe, C. T.; Ricks, M. J.; Siddall, T. L.; Yerkes, C. N.; Zhu, Y. U.S. Patent Application 2006/0089370.

4. Antifungal activities of novel non-azole molecules against S. cerevisiae and C. albicans

5. Babu, Y.; Chand, P.; Wu, M.; Kotian, P. L.; Kumar, V. S.; Lin, T.-H.; El-Kattan, Y.; Ghosh, A. K. WO 2006/050161.

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