Straightforward hit identification approach in fragment-based discovery of bromodomain-containing protein 4 (BRD4) inhibitors-Reference-Cited by-同舟云学术

Straightforward hit identification approach in fragment-based discovery of bromodomain-containing protein 4 (BRD4) inhibitors

Published:2018-07 Issue:12 Volume:26 Page:3399-3405
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Borysko Petro,Moroz Yurii S.,Vasylchenko Oleksandr V.,Hurmach Vasyl V.,Starodubtseva Anastasia,Stefanishena Natalia,Nesteruk Kateryna^ORCID,Zozulya Sergey,Kondratov Ivan S.,Grygorenko Oleksandr O.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference56 articles.

1. Erlanson DA, Jahnke W. In: Hubbard RE. (Ed.) Fragment-based Drug Discovery: Lessons and Outlook. Wiley-VCH Verlag GmbH & Co. KGaA, 2016; pp. 1–36.

2. What is the future for fragment-based drug discovery?

3. Fragments: past, present and future

4. Vemurafenib: the first drug approved for BRAF-mutant cancer

5. Venetoclax: A First-in-Class Oral BCL-2 Inhibitor for the Management of Lymphoid Malignancies

Cited by 16 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Fragment-based drug discovery for disorders of the central nervous system: designing better drugs piece by piece;Frontiers in Chemistry;2024-04-18

2. Target-based drug discovery: Applications of fluorescence techniques in high throughput and fragment-based screening;Heliyon;2024-01

3. Discovery of Small-Molecule TIM-3 Inhibitors for Acute Myeloid Leukemia Using Pharmacophore-Based Virtual Screening;Journal of Medicinal Chemistry;2023-08-11

4. Discovery of First-in-Class Small Molecule Inhibitors of Lymphocyte Activation Gene 3 (LAG-3);ACS Medicinal Chemistry Letters;2023-04-11

5. BET–HDAC Dual Inhibitors for Combinational Treatment of Breast Cancer and Concurrent Candidiasis;Journal of Medicinal Chemistry;2023-01-09