Structure based drug design and in vitro metabolism study: Discovery of N-(4-methylthiophenyl)-N,2-dimethyl-cyclopenta[d]pyrimidine as a potent microtubule targeting agent-Reference-Cited by-同舟云学术

Structure based drug design and in vitro metabolism study: Discovery of N-(4-methylthiophenyl)-N,2-dimethyl-cyclopenta[d]pyrimidine as a potent microtubule targeting agent

Published:2018-05 Issue:9 Volume:26 Page:2437-2451
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Xiang Weiguo,Choudhary Shruti,Hamel Ernest,Mooberry Susan L.,Gangjee Aleem

Funder

National Institutes of Health

National Cancer Institute

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

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5. Determinants of paclitaxel uptake, accumulation and retention in solid tumors;Jang;Invest New Drugs,2001

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