The 3-D conformational shape of N-naphthyl-cyclopenta[d]pyrimidines affects their potency as microtubule targeting agents and their antitumor activity-Reference-Cited by-同舟云学术

The 3-D conformational shape of N-naphthyl-cyclopenta[d]pyrimidines affects their potency as microtubule targeting agents and their antitumor activity

Published:2021-01 Issue: Volume:29 Page:115887
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Xiang Weiguo,Quadery Tasdique M.,Hamel Ernest^ORCID,Luckett-Chastain Lerin R.,Ihnat Michael A.^ORCID,Mooberry Susan L.,Gangjee Aleem

Funder

National Institutes of Health

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference35 articles.

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4. Microtubule destabilising agents: far more than just antimitotic anticancer drugs;Bates;Br J Clin Pharmacol,2017

5. Microtubule-targeting drugs: more than antimitotics;Kaul;J Nat Prod,2019

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