Overcoming HERG affinity in the discovery of the CCR5 antagonist maraviroc-Reference-Cited by-同舟云学术

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Overcoming HERG affinity in the discovery of the CCR5 antagonist maraviroc

Published:2006-09 Issue:17 Volume:16 Page:4633-4637
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Price David A.,Armour Duncan,de Groot Marcel,Leishman Derek,Napier Carolyn,Perros Manos,Stammen Blanda L.,Wood Anthony

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference12 articles.

1. The impact of drug-induced QT interval prolongation on drug discovery and development

2. Molecular and Cellular Mechanisms of Cardiac Arrhythmias

3. Antagonists of human CCR5 receptor containing 4-(pyrazolyl)piperidine side chains. Part 3: SAR studies on the benzylpyrazole segment

4. Greengrass, P. M.; Stewart, M.; Wood, C. M.; Patent Application WO 03021271.

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