Design, synthesis, and evaluation of JTE-013 derivatives as novel potent S1PR2 antagonists for recovering the sensitivity of colorectal cancer to 5-fluorouracil-Reference-Cited by-同舟云学术

Design, synthesis, and evaluation of JTE-013 derivatives as novel potent S1PR2 antagonists for recovering the sensitivity of colorectal cancer to 5-fluorouracil

Published:2023-02 Issue: Volume:131 Page:106318
ISSN:0045-2068
Container-title:Bioorganic Chemistry
language:en
Short-container-title:Bioorganic Chemistry

Author:

Guo Zhikun,Zhang Shuai,Liu Xiaochun,Zhao Guangjian,Zhang Yingzhi,Luo Dongdong,Zhao Xuecui,Xu Ximing,Qu Xianjun,Li Lin,Wan Shengbiao,Cui Shuxiang

Funder

National Natural Science Foundation of China

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

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3. S1PR2 Deficiency in DLBCL: a FOXy Connection;Baldari;Blood,2016

4. CD4 T Cell Sphingosine 1-Phosphate Receptor (S1PR)1 and S1PR4 and Endothelial S1PR2 Regulate Afferent Lymphatic Migration;Xiong;Sci. Immunol.,2019

5. Critical role of sphingosine-1-phosphate receptor 2 (S1PR2) in acute vascular inflammation;Zhang;Blood,2013

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