Design, synthesis, cyclooxygenase inhibition and biological evaluation of new 1,3,5-triaryl-4,5-dihydro-1 H -pyrazole derivatives possessing amino/methanesulfonyl pharmacophore-Reference-Cited by-同舟云学术

Design, synthesis, cyclooxygenase inhibition and biological evaluation of new 1,3,5-triaryl-4,5-dihydro-1 H -pyrazole derivatives possessing amino/methanesulfonyl pharmacophore

Published:2017-02 Issue: Volume:70 Page:57-66
ISSN:0045-2068
Container-title:Bioorganic Chemistry
language:en
Short-container-title:Bioorganic Chemistry

Author:

Abdellatif Khaled R.A.,Fadaly Wael A.A.

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

Reference30 articles.

1. Synthesis, biological evaluation and molecular modeling study of 5-trifluoromethyl-Δ2-pyrazoline and isomeric 5/3-trifluoromethylpyrazole derivatives as anti-inflammatory agents;Aggarwal;Eur. J. Med. Chem.,2013

2. Synthesis and anti-inflammatory activity of some novel 1,2-pyrazoline Derivatives;Gonjare;Der Pharma. Chemica.,2013

3. 2-Pyridinyl-3-(4-methylsulfonyl)phenylpyridines: selective and orally active cyclooxygenase-2 inhibitors;Friesen;Bioorg. Med. Chem. Lett.,1998

4. Pyridazinones as selective cyclooxygenase-2 inhibitors;Li;Bioorg. Med. Chem. Lett.,2003

5. Synthesis and anti-inflammatory activity of some new 1,3,5-trisubstituted pyrazolines bearing benzene sulfonamide;Rantish;Bioorg. Med. Chem. Lett.,2009

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