A novel derivatives of thiazol-4(5H)-one and their activity in the inhibition of 11β-hydroxysteroid dehydrogenase type 1
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry
Reference22 articles.
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3. The discovery of 2-anilinothiazolones as 11β-HSD1 inhibitors;Yuan;Bioorg. Med. Chem. Lett.,2007
4. 2-(S)-Phenethylaminothiazolones as potent, orally efficacious inhibitors of 11β-hydroxysteriod dehydrogenase type 1;Jean;J. Med. Chem.,2007
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1. Synthesis, characterization and biological activities of novel mononuclear nickel(II), copper(II) and chromium(III) complexes with N,N-dilaurylsubstituted thiazolidine-4-one-5-acetic acid ligand;2024-06-14
2. Synthesis, anti-diabetic profiling and molecular docking studies of 2-(2-arylidenehydrazinyl)thiazol-4(5 H )-ones;Future Medicinal Chemistry;2024-05-10
3. Lipophilic Studies and In Silico ADME Profiling of Biologically Active 2-Aminothiazol-4(5H)-one Derivatives;International Journal of Molecular Sciences;2023-07-31
4. Synthesis of Novel 2-(Cyclopentylamino)thiazol-4(5H)-one Derivatives with Potential Anticancer, Antioxidant, and 11β-HSD Inhibitory Activities;International Journal of Molecular Sciences;2023-04-14
5. 11β-Hydroxysteroid Dehydrogenase Type 1 as a Potential Treatment Target in Cardiovascular Diseases;Journal of Clinical Medicine;2022-10-20
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