Trifluoroethoxy group as a leaving group for regioselective sequential substitution reactions of 5-trifluoromethylpyrimidine derivative with heteroatom nucleophiles-Reference-Cited by-同舟云学术

Trifluoroethoxy group as a leaving group for regioselective sequential substitution reactions of 5-trifluoromethylpyrimidine derivative with heteroatom nucleophiles

Published:2015-11 Issue: Volume:179 Page:150-158
ISSN:0022-1139
Container-title:Journal of Fluorine Chemistry
language:en
Short-container-title:Journal of Fluorine Chemistry

Author:

Kagawa Takumi^ORCID,Shigehiro Daiki,Kawada Kosuke

Publisher

Elsevier BV

Subject

Inorganic Chemistry,Organic Chemistry,Physical and Theoretical Chemistry,Environmental Chemistry,Biochemistry

Reference21 articles.

1. The Lab Oddity Prevails: Discovery of Pan-CDK Inhibitor (R)-S-Cyclopropyl-S-(4-{[4-{[(1R,2R)-2-hydroxy-1-methylpropyl]oxy}-5-(trifluoromethyl)pyrimidin-2-yl]amino}phenyl)sulfoximide (BAY 1000394) for the Treatment of Cancer

2. New Pyrimidine Derivatives possessing ALK Inhibitory Activities

3. Sulfoximine-substituted trifluoromethylpyrimidine analogs as inhibitors of proline-rich tyrosine kinase 2 (PYK2) show reduced hERG activity

4. Discovery of Selective LRRK2 Inhibitors Guided by Computational Analysis and Molecular Modeling

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2. 2,2,2-Trifluoroethoxy Aromatic Heterocycles: Hydrolytically Stable Alternatives to Heteroaryl Chlorides;The Journal of Organic Chemistry;2018-10-19

3. Copper-Promoted Ritter-Type Trifluoroethoxylation of (Hetero)arenediazonium Tetrafluoroborates: A Method for the Preparation of Trifluoroethyl Imidates;European Journal of Organic Chemistry;2016-09-23