Successful Prediction of Human Pharmacokinetics After Oral Administration by Optimized Physiologically Based Pharmacokinetics Approach and Permeation Assay Using Human Induced Pluripotent Stem Cell–Derived Intestinal Epithelial Cells-Reference-Cited by-同舟云学术

Successful Prediction of Human Pharmacokinetics After Oral Administration by Optimized Physiologically Based Pharmacokinetics Approach and Permeation Assay Using Human Induced Pluripotent Stem Cell–Derived Intestinal Epithelial Cells

Published:2020-04 Issue:4 Volume:109 Page:1605-1614
ISSN:0022-3549
Container-title:Journal of Pharmaceutical Sciences
language:en
Short-container-title:Journal of Pharmaceutical Sciences

Author:

Mayumi Kei,Akazawa Takanori,Kanazu Takushi,Ohnishi Shuichi,Hasegawa Hiroshi

Publisher

Elsevier BV

Subject

Pharmaceutical Science

Reference73 articles.

1. The successes and failures of physiologically based pharmacokinetic modeling: there is room for improvement;Poggesi;Expert Opin Drug Metab Toxicol,2014

2. Successful prediction of human pharmacokinetics by improving calculation processes of physiologically based pharmacokinetic approach;Mayumi;J Pharm Sci,2019

3. In vitro-in vivo extrapolation of clearance: modeling hepatic metabolic clearance of highly bound drugs and comparative assessment with existing calculation methods;Poulin;J Pharm Sci,2012

4. Toward a new paradigm for the efficient in vitro-in vivo extrapolation of metabolic clearance in humans from hepatocyte data;Poulin;J Pharm Sci,2013

5. Prediction of the disposition of nine weakly acidic and six weakly basic drugs in humans from pharmacokinetic parameters in rats;Sawada;J Pharmacokinet Biopharm,1985

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