Simultaneous in-vivo receptor occupancy assays for serotonin 1A, 2A, and dopamine 2 receptors with the use of non-radiolabelled tracers: Proposed method in screening antipsychotics-Reference-Cited by-同舟云学术

Simultaneous in-vivo receptor occupancy assays for serotonin 1A, 2A, and dopamine 2 receptors with the use of non-radiolabelled tracers: Proposed method in screening antipsychotics

Published:2017-05 Issue: Volume:85 Page:22-28
ISSN:1056-8719
Container-title:Journal of Pharmacological and Toxicological Methods
language:en
Short-container-title:Journal of Pharmacological and Toxicological Methods

Author:

Thentu Jagadeesh Babu,Nirogi Ramakrishna,Bhyrapuneni Gopinadh,Ajjala Devender Reddy,Aleti Raghupathi Reddy,Palacharla Raghava Choudary

Funder

Suven Life Sciences Ltd.

Publisher

Elsevier BV

Subject

Pharmacology,Toxicology

Reference28 articles.

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3. Comparison of in vivo receptor occupancy studies using a radioligand-based approach or a liquid chromatography/mass spectrometry - based approach;Cao,2016

4. Antipsychotic drugs, neurotransmitters, and schizophrenia;Carlsson;The American Journal of Psychiatry,1978

5. Use of LC/MS to assess brain tracer distribution in preclinical, in vivo receptor occupancy studies: Dopamine D2, serotonin 2A and NK-1 receptor as examples;Chernet;Life Sciences,2005

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