Hypoxia-inducible factor inhibitors: a survey of recent patented compounds (2004 – 2010)
Author:
Publisher
Informa Healthcare
Subject
Drug Discovery,Pharmacology,General Medicine
Link
http://www.tandfonline.com/doi/pdf/10.1517/13543776.2011.547477
Reference66 articles.
1. A nuclear factor induced by hypoxia via de novo protein synthesis binds to the human erythropoietin gene enhancer at a site required for transcriptional activation.
2. Vascular endothelial growth factor induced by hypoxia may mediate hypoxia-initiated angiogenesis
3. Hypoxia-inducible factor 1 is a basic-helix-loop-helix-PAS heterodimer regulated by cellular O2 tension.
4. Identification of the von Hippel-Lindau tumor-suppressor protein as part of an active E3 ubiquitin ligase complex
5. The tumour suppressor protein VHL targets hypoxia-inducible factors for oxygen-dependent proteolysis
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