Design, synthesis, and evaluation of indeno[2,1-c]pyrazolones for use as inhibitors against hypoxia-inducible factor (HIF)-1 transcriptional activity-Reference-Cited by-同舟云学术

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Design, synthesis, and evaluation of indeno[2,1-c]pyrazolones for use as inhibitors against hypoxia-inducible factor (HIF)-1 transcriptional activity

Published:2020-01 Issue:1 Volume:28 Page:115207
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Fuse Shinichiro,Suzuki Kensuke,Kuchimaru Takahiro,Kadonosono Tetsuya,Ueda Hiroki,Sato Shinichi,Kizaka-Kondoh Shinae,Nakamura Hiroyuki

Funder

Ministry of Education, Culture, Sports, Science and Technology, Japan

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference54 articles.

1. Hypoxia-inducible factor 1 is a basic-helix-loop-helix-PAS heterodimer regulated by cellular O2 tension.

2. Dimerization, DNA Binding, and Transactivation Properties of Hypoxia-inducible Factor 1

3. A Conserved Family of Prolyl-4-Hydroxylases That Modify HIF

4. C. elegans EGL-9 and Mammalian Homologs Define a Family of Dioxygenases that Regulate HIF by Prolyl Hydroxylation

5. The tumour suppressor protein VHL targets hypoxia-inducible factors for oxygen-dependent proteolysis

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