Synthesis and identification of GZD856 as an orally bioavailable Bcr-AblT315I inhibitor overcoming acquired imatinib resistance
Author:
Affiliation:
1. School of Pharmacy, Jinan University, Guangzhou, China;
2. State Key Laboratory of Respiratory Diseases, Guangzhou Institutes of Biomedicine and Health, Chinese Academy of Sciences, Guangzhou, China
Funder
National High Technology Research and Development
Guangdong Natural Science Funds for Distinguished Young Scholar
Pearl River S&T Nova Program of Guangzhou
Guangdong Special Branch Program Technology Young Talents
Publisher
Informa UK Limited
Subject
Drug Discovery,Pharmacology,General Medicine
Link
https://tandfonline.com/doi/pdf/10.1080/14756366.2016.1250757
Reference29 articles.
1. A New Consistent Chromosomal Abnormality in Chronic Myelogenous Leukaemia identified by Quinacrine Fluorescence and Giemsa Staining
2. Molecular biology of bcr-abl1–positive chronic myeloid leukemia
3. Glivec (STI571, imatinib), a rationally developed, targeted anticancer drug
4. The development of imatinib as a therapeutic agent for chronic myeloid leukemia
5. Imatinib and beyond—exploring the full potential of targeted therapy for CML
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